Characterization of an Akt Kinase Inhibitor with Potent Pharmacodynamic and Antitumor Activity Dirk A. Heerding, Derek R. Duckett, et al. Cancer Res 2008;68:2366-2374
Identification of 4-(2-(4-Amino-1,2,5-oxadiazol-3-yl)-1-ethyl-7-{[(3S)-3-piperidinylmethyl]oxy}-1H-imidazo[4,5-c]pyridin-4-yl)-2-methyl-3-butyn-2-ol (GSK690693), a Novel Inhibitor of AKT Kinase Dirk A. Heerding,Nelson Rhodes,et al. J. Med. Chem 2008;51: 5663–5679
The pharmacological and toxicological properties of this product have not been fully investigated. Exercise caution in use and handling. This product must not be used in humans.